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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $211.65 | Total: $1,058.25 |
| 1 | 10 | $179.28 | Total: $1,792.80 |
| 1 | 25 | $151.89 | Total: $3,797.25 |
| 1 | 50 | $129.48 | Total: $6,474.00 |
| 1 | 100 | $112.05 | Total: $11,205.00 |
Overview
Sarizotan HCl (EMD 128130 HCl) is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinson's Dyskinesia.
Chemical Properties
| Molecular Formula | C22H22ClFN2O |
| Molecular Weight | 384.87 |
| CAS Numbers | 195068-07-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(NC[C@@H]1OC=2C(CC1)=CC=CC2)C3=CC(=CN=C3)C4=CC=C(F)C=C4.Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Cheng H,et al. Potent hERG channel inhibition by sarizotan, an investigative treatment for Rett Syndrome. J Mol Cell Cardiol. 2019 Oct;135 22-30.