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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $166.60 | Total: $833.00 |
| 1 | 10 | $141.12 | Total: $1,411.20 |
| 1 | 25 | $119.56 | Total: $2,989.00 |
| 1 | 50 | $101.92 | Total: $5,096.00 |
| 1 | 100 | $88.20 | Total: $8,820.00 |
Overview
Naluzotan hydrochloride (PRX 00023 hydrochloride) is a hERG K+ channel blocker with an IC50 value of 3800 nM and is commonly used in the study of anxiety and depression.Naluzotan hydrochloride is also a novel, potent, and selective 5-HT1A agonist, with an IC50 value of about 20 nM and a Ki value of about 5.1 Naluzotan hydrochloride is also a novel, potent and selective 5-HT1A agonist with an IC50 of approximately 20 nM and a Ki of approximately 5.1 nM.
Chemical Properties
| Molecular Formula | C23H39ClN4O3S |
| Molecular Weight | 487.1 |
| CAS Numbers | 740873-82-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.O=C(NC1=CC=CC(=C1)N2CCN(CC2)CCCCNS(=O)(=O)CC3CCCCC3)C |
Storage and Handling
0C Short Term, -20C Long Term
References
Becker OM, et al. An integrated in silico 3D model-driven discovery of a novel, potent, and selective amidosulfonamide 5-HT1A agonist [PRX-00023] for the treatment of anxiety and depression. J Med Chem. 2006 Jun 1;49[11] 3116-35.