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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $141.10 | Total: $705.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 100 | $74.70 | Total: $7,470.00 |
Overview
Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.
Chemical Properties
| Molecular Formula | C19H21FN2O2 |
| Molecular Weight | 328.38 |
| CAS Numbers | 130579-75-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)CCON=C(C=Cc1ccc(O)cc1)c1ccccc1F |
Storage and Handling
0C Short Term, -20C Long Term
References
Malgorzata Filip, et al. Contribution of serotonin [5-hydroxytryptamine; 5-HT] 5-HT2 receptor subtypes to the hyperlocomotor effects of cocaine acute and chronic pharmacological analyses. J Pharmacol Exp Ther. 2004 Sep;310[3] 1246-54.