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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $59.50 | Total: $297.50 |
| 1 | 10 | $50.40 | Total: $504.00 |
| 1 | 25 | $42.70 | Total: $1,067.50 |
| 1 | 50 | $36.40 | Total: $1,820.00 |
| 1 | 100 | $31.50 | Total: $3,150.00 |
Overview
BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.
Chemical Properties
| Molecular Formula | C19H27ClN4O2 |
| Molecular Weight | 378.9 |
| CAS Numbers | 134296-40-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.CC(C)n1c2ccccc2n(C(=O)N[C@@H]2C[C@@H]3CC[C@H](C2)N3C)c1=O |
Storage and Handling
0C Short Term, -20C Long Term
References
H Pan , et al. 5-HT1A and 5-HT4 receptors mediate inhibition and facilitation of fast synaptic transmission in enteric neurons. Am J Physiol. 1994 Feb;266[2 Pt 1] G230-8.