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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $39.95 | Total: $199.75 |
| 1 | 10 | $33.84 | Total: $338.40 |
| 1 | 25 | $28.67 | Total: $716.75 |
| 1 | 50 | $24.44 | Total: $1,222.00 |
| 1 | 100 | $21.15 | Total: $2,115.00 |
Overview
LY 272015 hydrochloride is an orally active and selective 5-HT2B receptor antagonist that displays antihypertensive effects in DOCA-salt hypertensive rats.LY 272015 hydrochloride inhibits 5-HT- or BW723C86-induced ERK2 phosphorylation and attenuates MVIC and Tissue downstream cellular effects of 5HT signaling and can be used to study hepatocellular carcinoma.
Chemical Properties
| Molecular Formula | C21H25ClN2O2 |
| Molecular Weight | 372.89 |
| CAS Numbers | 172895-15-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.O(C1=CC=C(C=C1OC)CC2NCCC=3C=4C=C(C=CC4NC32)C)C |
Storage and Handling
0C Short Term, -20C Long Term
References
Russell A, et al. 5-Hydroxytryptamine[2B] receptor function is enhanced in the N[omega]-nitro-L-arginine hypertensive rat. J Pharmacol Exp Ther. 2002 Oct;303[1] 179-87.