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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $29.75 | Total: $148.75 |
| 1 | 10 | $25.20 | Total: $252.00 |
| 1 | 25 | $21.35 | Total: $533.75 |
| 1 | 50 | $18.20 | Total: $910.00 |
| 1 | 100 | $15.75 | Total: $1,575.00 |
Overview
SB 258585 is a selective 5-HT6 receptor antagonist.SB 258585 has a high affinity for individual receptor populations in cell lines with human recombinant 5-HT6 receptors.SB 258585 can be used to label both recombinant and natural 5-HT6 receptors, and can be used to assay cognitive enhancement and antipsychotic activity.
Chemical Properties
| Molecular Formula | C18H22IN3O3S |
| Molecular Weight | 487.36 |
| CAS Numbers | 209480-63-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=S(NC1=CC=C(C(N2CCN(CC2)C)=C1)OC)(C3=CC=C(C=C3)I)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Hirst WD, et al. Characterization of [[125]I]-SB-258585 binding to human recombinant and native 5-HT[6] receptors in rat, pig and human brain tissue. Br J Pharmacol. 2000 Aug;130[7] 1597-605.