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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $58.65 | Total: $293.25 |
| 1 | 10 | $49.68 | Total: $496.80 |
| 1 | 25 | $42.09 | Total: $1,052.25 |
| 1 | 50 | $35.88 | Total: $1,794.00 |
| 1 | 100 | $31.05 | Total: $3,105.00 |
Overview
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM). Facinicline hydrochloride improves cognition and sensorimotor gating in rodents.
Chemical Properties
| Molecular Formula | C15H19ClN4O |
| Molecular Weight | 306.79 |
| CAS Numbers | 677305-02-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.O=C(N[C@@H]1CN2CCC1CC2)c1n[nH]c2ccccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Boess F, et al. Use of early phenotypic in vivo markers to assess human relevance of an unusual rodent non-genotoxic carcinogen in vitro. Toxicology. 2017 Mar 15;379 48-61.