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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380
Chemical Properties
| Molecular Formula | C18H19N3O2S |
| Molecular Weight | 341.43 |
| CAS Numbers | 409351-28-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1ccc(CNC(=O)c2sc3nc(C)cc(C)c3c2N)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Brady AE, et al. Centrally active allosteric potentiators of the M4 muscarinic acetylcholine receptor reverse amphetamine-induced hyperlocomotor activity in rats. J Pharmacol Exp Ther. 2008 Dec;327[3] 941-53.