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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $39.10 | Total: $195.50 |
| 1 | 10 | $33.12 | Total: $331.20 |
| 1 | 25 | $28.06 | Total: $701.50 |
| 1 | 50 | $23.92 | Total: $1,196.00 |
| 1 | 100 | $20.70 | Total: $2,070.00 |
Overview
Centanafadine hydrochloride (EB-1020 hydrochloride) is a dual inhibitor of norepinephrine (NE)dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83 nM for human NE, DA, and serotonin transporter).
Chemical Properties
| Molecular Formula | C15H16ClN |
| Molecular Weight | 245.75 |
| CAS Numbers | 923981-14-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.C1[C@@H]2CNC[C@]12c1ccc2ccccc2c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Bymaster FP, et al. Pharmacological characterization of the norepinephrine and dopamine reuptake inhibitor EB-1020 implications for treatment of attention-deficit hyperactivity disorder. Synapse. 2012 Jun;66[6] 522-32.