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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $96.05 | Total: $480.25 |
| 1 | 10 | $81.36 | Total: $813.60 |
| 1 | 25 | $68.93 | Total: $1,723.25 |
| 1 | 50 | $58.76 | Total: $2,938.00 |
| 1 | 100 | $50.85 | Total: $5,085.00 |
Overview
Lusaperidone (R107474) is a potent ?2-adrenergic receptor antagonist, a potential radioligand for the ? (2)-adrenergic receptor, with inhibitory effects on ?2A and ?2C, with Ki values of 0.13 and 0.15 nM, respectively.
Chemical Properties
| Molecular Formula | C22H21N3O2 |
| Molecular Weight | 359.42 |
| CAS Numbers | 214548-46-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1nc2ccccn2c(=O)c1CCN1CCc2oc3ccccc3c2C1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Van der Mey M, et al. Synthesis and biodistribution of [11C]R107474, a new radiolabeled alpha2-adrenoceptor antagonist. Bioorg Med Chem. 2006 Jul 1;14[13] 4526-34.