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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Overview
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (?2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a Kb value (antagonist activity) of 16 nM.
Chemical Properties
| Molecular Formula | C24H26Cl2N4 |
| Molecular Weight | 441.4 |
| CAS Numbers | 1259314-65-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cl.CN1CCN(CC1)c1ccc(Nc2c3ccccc3nc3ccccc23)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Tricklebank MD, et al. JP-1302 a new tool to shed light on the roles of alpha2C-adrenoceptors in brain. Br J Pharmacol. 2007 Feb;150[4] 381-2.