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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $80.75 | Total: $403.75 |
| 1 | 10 | $68.40 | Total: $684.00 |
| 1 | 25 | $57.95 | Total: $1,448.75 |
| 1 | 50 | $49.40 | Total: $2,470.00 |
| 1 | 100 | $42.75 | Total: $4,275.00 |
Overview
Fezolamine is a novel orally available non-tricyclic compound with antidepressant activity. It is three to two times more selective in blocking synaptosomal uptake of [3H]norepinephrine than uptake of [4H]3-hydroxytryptamine or [3H]dopamine in vitro. It blocked the inhibitory effects of rifampicin and tetraphenyl in classical behavioral tests using monoamine-depleted animals.
Chemical Properties
| Molecular Formula | C20H23N3 |
| Molecular Weight | 305.42 |
| CAS Numbers | 80410-36-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(CCN(C)C)N1C=C(C(=N1)C2=CC=CC=C2)C3=CC=CC=C3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Zisook S, et al. Efficacy and safety of fezolamine in depressed patients. Neuropsychobiology. 1987;17[3] 133-138.