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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $113.90 | Total: $569.50 |
| 1 | 10 | $96.48 | Total: $964.80 |
| 1 | 25 | $81.74 | Total: $2,043.50 |
| 1 | 50 | $69.68 | Total: $3,484.00 |
| 1 | 100 | $60.30 | Total: $6,030.00 |
Overview
Saterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular ?-1-adrenoceptor. Saterinone has vasodilatory properties and can be used in the acute treatment of chronic heart failure. Saterinone inhibited crude cAMP phosphodiesterase (PDE) activity in guinea pig right ventricular homogenates The ic50 value is 2.3
Chemical Properties
| Molecular Formula | C27H30N4O4 |
| Molecular Weight | 474.55 |
| CAS Numbers | 102669-89-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC1=C(C=C(C#N)C(=O)N1)C2=CC=C(OCC(CN3CCN(CC3)C4=C(OC)C=CC=C4)O)C=C2 |
Storage and Handling
0C Short Term, -20C Long Term
References
Brunkhorst D, et al. Selective inhibition of cAMP phosphodiesterase III activity by the cardiotonic agent saterinone in guinea pig myocardium. Arzneimittelforschung. 1988;38[9] 1293-1298.