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View larger CB1 inverse agonist 1
AT10694
CAS 852315-00-5
Molarity Calculation Cart®
HOW TO ORDER
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $44.55 | Total: $4,455.00 |
| 1 | 50 | $51.48 | Total: $2,574.00 |
| 1 | 25 | $60.39 | Total: $1,509.75 |
| 1 | 10 | $71.28 | Total: $712.80 |
| 1 | 5 | $84.15 | Total: $420.75 |
Data sheet
| Molecular Formula | C25H18Cl3N3O3 |
| Molecular Weight | 514.79 |
| CAS Numbers | 852315-00-5 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C(C)=O)C=1C=2C(=NC(=C(C2)C3=CC=C(Cl)C=C3)C4=C(Cl)C=C(Cl)C=C4)N(C)C(=O)C1C(C)=O |
| References | Debenham JS, et al. Synthesis of functionalized 1,8-naphthyridinones and their evaluation as novel, orally active CB1 receptor inverse agonists.Bioorg Med Chem Lett. 2006 Feb;16[3] 681-5. |
More info
CB1 inverse agonist 1 (MRL-650) is an orally active and selective CB1 agonist. The IC50s for CB1 and CB2 are 7.5 nM and 4100 nM, respectively. CB1 inverse agonist 1 shows anorexigenic effects.