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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $164.90 | Total: $824.50 |
| 1 | 10 | $139.68 | Total: $1,396.80 |
| 1 | 25 | $118.34 | Total: $2,958.50 |
| 1 | 50 | $100.88 | Total: $5,044.00 |
| 1 | 100 | $87.30 | Total: $8,730.00 |
Overview
PXS-6302 hydrochloride is a potent irreversible lysine oxidase (LOX) inhibitor, inhibiting Bovine LOX, rh LOXL1, rh LOXL2, rh LOXL3, and rh LOXL4 with IC50 of 3.7 ?M, 3.4 ?M, 0.4 ?M, 1.5 ?M, and 0.3 ?M, respectively. PXS-6302 hydrochloride penetrates easily through the skin and is able to reduce collagen accumulation, significantly improving the appearance of scars.
Chemical Properties
| Molecular Formula | C10H11ClF3NO2S |
| Molecular Weight | 301.71 |
| CAS Numbers | 2584947-79-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | S(C(C(=CCN)F)(F)F)(=O)(=O)C1=CC=CC=C1.Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Chaudhari N, et al. Topical application of an irreversible small molecule inhibitor of lysyl oxidases ameliorates skin scarring and fibrosis. Nat Commun. 2022 Sep 22;13[1] 5555.