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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $60.35 | Total: $301.75 |
| 1 | 10 | $51.12 | Total: $511.20 |
| 1 | 25 | $43.31 | Total: $1,082.75 |
| 1 | 50 | $36.92 | Total: $1,846.00 |
| 1 | 100 | $31.95 | Total: $3,195.00 |
Overview
Nampt activator-2 is a NAMPT activator (EC50: 0.023 ?M). Nampt activator-2 has an affinity for CYP2C9, 2D6, and 2C19 with affinity values of 0.060 ?M, 0.41 ?M, and 0.59 ?M, respectively.Nampt activator-2 can be used in the study of atherosclerosis, obesity, type II diabetes, insulin resistance, and type I diabetes.
Chemical Properties
| Molecular Formula | C17H15ClN4O3S |
| Molecular Weight | 390.84 |
| CAS Numbers | 2237268-90-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | S(=O)(=O)(C1=CC=C(NC(NCC=2C=NNC2)=O)C=C1)C3=CC=C(Cl)C=C3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Pinkerton AB, et al. Optimization of a urea-containing series of nicotinamide phosphoribosyltransferase [NAMPT] activators. Bioorg Med Chem Lett. 2021 Jun 1;41 128007.