Categories
- PROTAC Linker
- Protein Control Ligand
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $25.50 | Total: $127.50 |
| 1 | 10 | $21.60 | Total: $216.00 |
| 1 | 25 | $18.30 | Total: $457.50 |
| 1 | 50 | $15.60 | Total: $780.00 |
| 1 | 100 | $13.50 | Total: $1,350.00 |
Overview
GLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.
Chemical Properties
| Molecular Formula | C24H21NO3 |
| Molecular Weight | 371.43 |
| CAS Numbers | 421578-93-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC1(CC(=O)c2ccccc2)C(=O)N(CCc2ccccc2)c2ccccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Wang J, et al. Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site. ACS Chem Biol. 2021 Nov 19;16[11] 2444-2452.