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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $50.15 | Total: $250.75 |
| 1 | 10 | $42.48 | Total: $424.80 |
| 1 | 25 | $35.99 | Total: $899.75 |
| 1 | 50 | $30.68 | Total: $1,534.00 |
| 1 | 100 | $26.55 | Total: $2,655.00 |
Overview
Epitinib succinate (HMPL-813 succinate) is an orally active and brain penetration EGFR tyrosine kinase inhibitor and can be used in studies about cancer.
Chemical Properties
| Molecular Formula | C28H32N6O6 |
| Molecular Weight | 548.59 |
| CAS Numbers | 2252334-12-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC(=O)CCC(O)=O.CCN1CCN(CC1)C(=O)Nc1cc2c(Nc3cccc(c3)C#C)ncnc2cc1OC |
Storage and Handling
0C Short Term, -20C Long Term
References
Zhou et al. The safety profile of a selective EGFR TKI epitinib [HMPL-813] in patients with advanced solid tumors and preliminary clinical efficacy in EGFRm+ NSCLC patients with brain metastasis. Journal of Clinical Oncology 2016 34 15_suppl, e20502-e20502