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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $103.70 | Total: $518.50 |
| 1 | 10 | $87.84 | Total: $878.40 |
| 1 | 25 | $74.42 | Total: $1,860.50 |
| 1 | 50 | $63.44 | Total: $3,172.00 |
| 1 | 100 | $54.90 | Total: $5,490.00 |
Overview
Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value for antagonism of histamine-induced positive chronotropic responses in the right atrium of isolate guinea pigs was 0.041.Dalcotidine improves the quality of ulcer healing, and may contribute to a reduction in ulcer recurrence and relapse rates.
Chemical Properties
| Molecular Formula | C18H29N3O2 |
| Molecular Weight | 319.44 |
| CAS Numbers | 120958-90-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(C1=CC(OCCCNC(NCC)=O)=CC=C1)N2CCCCC2 |
Storage and Handling
0C Short Term, -20C Long Term
References
Sekiguchi H, et al. Pharmacological profiles of the new histamine H2-receptor antagonist N-ethyl-N'-[3-[3-[piperidinomethyl]phenoxy] propyl] urea. Arzneimittelforschung. 1993;43[2] 129-133.