Histamine Receptors

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Enerisant

AT67828

CAS 1152747-82-4

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$83.00

$83.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $37.35 Total: $3,735.00
150 $43.16 Total: $2,158.00
125 $50.63 Total: $1,265.75
110 $59.76 Total: $597.60
15 $70.55 Total: $352.75

Data sheet

Molecular FormulaC22H30N4O3
Molecular Weight398.5
CAS Numbers1152747-82-4
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeC(=O)(C1=CN(N=C1)C2=CC=C(OCCCN3[C@H](C)CCC3)C=C2)N4CCOCC4
ReferencesHino N, et al. A novel potent and selective histamine H3 receptor antagonist enerisant in vitro profiles, in vivo receptor occupancy, and wake-promoting and procognitive effects in rodents. Journal of Pharmacology and Experimental Therapeutics, 2020, 375[2] 276-285.

More info

Enerisant (TS-091) is an orally active, selective and potent histamine H3 receptor antagonist that modulates histamine H3 receptors in mice in a dose-dependent manner.Enerisant promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.