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View larger PF-03654746
AT16476
CAS 935840-31-6
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $182.75 | Total: $913.75 |
| 1 | 10 | $154.80 | Total: $1,548.00 |
| 1 | 25 | $131.15 | Total: $3,278.75 |
| 1 | 50 | $111.80 | Total: $5,590.00 |
| 1 | 100 | $96.75 | Total: $9,675.00 |
Data sheet
| Molecular Formula | C18H24F2N2O |
| Molecular Weight | 322.39 |
| CAS Numbers | 935840-31-6 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | F[C@@]1(C[C@@H](C(NCC)=O)C1)C2=CC(F)=C(CN3CCCC3)C=C2 |
| References | Brioni JD, et al. Discovery of histamine H3 antagonists for the treatment of cognitive disorders and Alzheimer's disease. J Pharmacol Exp Ther. 2011 Jan;336[1] 38-46. |
More info
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease. PF-03654746 can be used in studies about the treatment of allergic rhinitis.