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View larger PF-03654764
AT61213
CAS 935840-35-0
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $237.15 | Total: $1,185.75 |
| 1 | 10 | $200.88 | Total: $2,008.80 |
| 1 | 25 | $170.19 | Total: $4,254.75 |
| 1 | 50 | $145.08 | Total: $7,254.00 |
| 1 | 100 | $125.55 | Total: $12,555.00 |
Data sheet
| Molecular Formula | C20H28F2N2O |
| Molecular Weight | 350.45 |
| CAS Numbers | 935840-35-0 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)CNC(=O)[C@H]1C[C@](F)(C1)c1ccc(CN2CCCC2)c(F)c1 |
| References | Michelle L North, et al. Add-on histamine receptor-3 antagonist for allergic rhinitis a double blind randomized crossover trial using the environmental exposure unit. Allergy Asthma Clin Immunol. 2014 Jul 3;10[1] 33. |
More info
PF-03654764 is an orally active, potent, and selective histamine H3 receptor antagonist with Ki values of 1.2 nM for human H3 and 7.9 nM for rat H3. It is often co-administered with Fexofenadine for the treatment of allergic rhinitis.