KCC2 - K-Cl co-transporter

Opiranserin hydrochloride View larger

Opiranserin hydrochloride

AT9833

CAS 1440796-75-7

More details

Molarity Calculation Cart®

HOW TO ORDER

$82.00

$82.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $36.90 Total: $3,690.00
150 $42.64 Total: $2,132.00
125 $50.02 Total: $1,250.50
110 $59.04 Total: $590.40
15 $69.70 Total: $348.50

Data sheet

Molecular FormulaC21H35ClN2O5
Molecular Weight430.97
CAS Numbers1440796-75-7
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCl.CCCCOc1c(OC)cc(cc1OC)C(=O)NCC1(CCOCC1)N(C)C

More info

Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 ?M, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 ?M). It is development as an injectable agent for the treatment of postoperative pain.