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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $69.70 | Total: $348.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 100 | $36.90 | Total: $3,690.00 |
Overview
Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 ?M, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 ?M). It is development as an injectable agent for the treatment of postoperative pain.
Chemical Properties
| Molecular Formula | C21H35ClN2O5 |
| Molecular Weight | 430.97 |
| CAS Numbers | 1440796-75-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.CCCCOc1c(OC)cc(cc1OC)C(=O)NCC1(CCOCC1)N(C)C |
Storage and Handling
0C Short Term, -20C Long Term