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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $135.15 | Total: $675.75 |
| 1 | 10 | $114.48 | Total: $1,144.80 |
| 1 | 25 | $96.99 | Total: $2,424.75 |
| 1 | 50 | $82.68 | Total: $4,134.00 |
| 1 | 100 | $71.55 | Total: $7,155.00 |
Overview
MBM-55 is an effective inhibitor of NIMA related kinase 2 (NEK2) with an IC50 of 1 nM. MBM-55 effectively inhibits the proliferation of cancer cells by inducing cell cycle arrest and apoptosis.
Chemical Properties
| Molecular Formula | C28H27FN6O2 |
| Molecular Weight | 498.55 |
| CAS Numbers | 2083622-09-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)CCn1cc(cn1)-c1ccn2c(cnc2c1)-c1ccc(C(N)=O)c(OCc2cccc(F)c2)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Xi JB, et al. Structure-based design and synthesis of imidazo[1,2-a]pyridine derivatives as novel and potent Nek2 inhibitors with in vitro and in vivo antitumor activities. Eur J Med Chem. 2017 Jan 27;126 1083-1106.