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Norketotifen hydrogen fumarate
AOB16140G
CAS: 930765-16-5
Chemical Name: 2-Piperidin-4-ylidene-6-thiatricyclo[8.4.0.03,7]tetradeca-1(14),3(7),4,10,12-pentaen-8-one hydrogen fumarate
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $31.05 | Total: $3,105.00 |
| 1 | 50 | $35.88 | Total: $1,794.00 |
| 1 | 25 | $42.09 | Total: $1,052.25 |
| 1 | 10 | $49.68 | Total: $496.80 |
| 1 | 5 | $58.65 | Total: $293.25 |
Data sheet
| Molecular Formula | C22H21NO5S |
| Molecular Weight | 411.47 |
| CAS Numbers | 930765-16-5 |
| Storage Condition | 0°C (short term), -20°C (long term), desiccated |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| Synonym | Norketotifen |
| IUPAC/Chemical Name | 2-Piperidin-4-ylidene-6-thiatricyclo[8.4.0.03,7]tetradeca-1(14),3(7),4,10,12-pentaen-8-one hydrogen fumarate |
| InChl Key | PDPPFVXCBONTQQ-WLHGVMLRSA-N |
| InChl Code | 1S/C18H17NOS.C4H4O4/c20-16-11-13-3-1-2-4-14(13)17(12-5-8-19-9-6-12)15-7-10-21-18(15)16;5-3(6)1-2-4(7)8/h1-4,7,10,19H,5-6,8-9,11H2;1-2H,(H,5,6)(H,7,8)/b;2-1+ |
| SMILES Code | c1ccc2c(c1)CC(=O)c3c(ccs3)C2=C4CCNCC4.C([H])(=C(/[H])C(=O)O)/C(=O)O |
| References | 1) Axel Karl Gunnar Aberg et al., Ketotifen is a Prodrug. Norketotifen is the active metabolite, Drug Dev Res., 2022 Apr;83(2):362-367. doi: 10.1002/ddr.21865. Epub 2021 Aug 19. |
| PubChem ID | 45489140 |
More info
The anti-inflammatory active metabolite of Ketotifen for the treatment of uncomplicated influenza-like illness