Neuropeptide Receptors

SB-222200 View larger

SB-222200

AT16849

CAS 174635-69-9

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$28.00

$28.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $12.60 Total: $1,260.00
150 $14.56 Total: $728.00
125 $17.08 Total: $427.00
110 $20.16 Total: $201.60
15 $23.80 Total: $119.00

Data sheet

Molecular FormulaC26H24N2O
Molecular Weight380.48
CAS Numbers174635-69-9
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeNc1cccc(CN2C(Cc3ccccc3)C(O)C(O)C(Cc3ccccc3)N(Cc3cccc(N)c3)C2=O)c1
ReferencesSarau HM, et al. Nonpeptide tachykinin receptor antagonists. II. Pharmacological and pharmacokinetic profile of SB-222200, a central nervous system penetrant, potent and selective NK-3 receptor antagonist. J Pharmacol Exp Ther. 2000 Oct;295[1] 373-81.

More info

SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).