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Opioid Receptors
- Protein Control Ligand
- Pathway Inhibitors
- Enzyme Inhibitors
- Kinase Inhibitors
- Protease
- Synthase
- p18
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- p70
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- Peptidase
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- Hydroxylases
- Ubiquitin-Activating Enzyme
- Adenosine Deaminase
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- p68
- ACE
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- Transferase
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- Cell Inhibition
- Synthase
- Receptor Tyrosine Phosphatases (RTP)
- AChE
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- Autophagy
- Toll-Like Receptor (TLR)
- Enzyme Inhibitors
- Function Modulators
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- G Protein-Coupled Receptor Ligands
- 5HT Receptors
- Adrenoceptor
- Angiotensin Receptor
- Cannabinoid Receptors
- CCK Receptors
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- Ghrelin Receptors
- GABA Receptors
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- Metabotropic Glutamate Receptors
- Motilin Receptors
- Muscarinic Receptor
- Neuropeptide Receptors
- Opioid Receptors
- Orexin Receptors
- Orphan Receptors
- Prostanoid Receptors
- Proteinase-Activated Receptors
- Purinergic Receptors
- Ryanodine receptor
- Sigma Receptors
- Thrombin Receptor
- Vaniloid Receptor
- VIP and PACAP Receptors
- Neurotensin Receptors
- Urotensin Receptor
- Imidazoline receptor
- SMO Receptors
- Apelin Receptor
- β-arrestin/β2-adaptin
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- CFTR
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- Biomarkers and Buffer Solutions
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- Customized Screening Library
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- Molecular Glues
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- SARS-CoV
View larger Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $44.55 | Total: $4,455.00 |
| 1 | 50 | $51.48 | Total: $2,574.00 |
| 1 | 25 | $60.39 | Total: $1,509.75 |
| 1 | 10 | $71.28 | Total: $712.80 |
| 1 | 5 | $84.15 | Total: $420.75 |
Data sheet
| Molecular Formula | C20H22ClN5 |
| Molecular Weight | 367.88 |
| CAS Numbers | 1174985-59-1 |
| Storage Condition | 0C Short Term, -20C Long Term |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC1=C(N(N=C1CNC2CCCC2)C3=C(Cl)C=CC=N3)C=4C=CC=NC4 |
| References | Kobayashi K, et al. Discovery of novel arylpyrazole series as potent and selective opioid receptor-like 1 [ORL1] antagonists. Bioorg Med Chem Lett. 2009 Jul 1;19[13] 3627-31. |
More info
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).