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> G Protein-Coupled Receptor Ligands>Opioid Receptors>Dynorphin A 1-10 acetate(79994-24-4 free base)

Opioid Receptors

Dynorphin A 1-10 acetate(79994-24-4 free base) View larger

Dynorphin A 1-10 acetate(79994-24-4 free base)

ATP1813L

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$86.00

$86.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $73.10 Total: $365.50
110 $61.92 Total: $619.20
125 $52.46 Total: $1,311.50
150 $44.72 Total: $2,236.00
1100 $38.70 Total: $3,870.00

Data sheet

Molecular FormulaC59H95N19O14
Molecular Weight1294.53
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeO=C([C@H](CCCNC(N)=N)NC([C@H]([C@@H](C)CC)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@@H](NC(CNC(CNC([C@@H](N)CC1=CC=C(O)C=C1)=O)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O)=O)N3[C@H](C(O)=O)CCC3.CC(O)=O
ReferencesPaterlini G, et al. Molecular simulation of dynorphin A-[1-10] binding to extracellular loop 2 of the kappa-opioidreceptor. A model for receptor activation. J Med Chem. 1997 Sep 26;40[20] 3254-62.

More info

Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the ?-opioid receptor. Dynorphin A (1-10) also blocks NMDA-activated current with an IC50 of 42.0 ?M.