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> G Protein-Coupled Receptor Ligands>Opioid Receptors>[(pF)Phe4]Nociceptin(1-13)NH2 acetate

Opioid Receptors

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[(pF)Phe4]Nociceptin(1-13)NH2 acetate

ATP1885L1

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$278.00

$278.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $236.30 Total: $1,181.50
110 $200.16 Total: $2,001.60
125 $169.58 Total: $4,239.50
150 $144.56 Total: $7,228.00
1100 $125.10 Total: $12,510.00

Data sheet

Molecular FormulaC63H103FN22O17
Molecular Weight1459.63
Storage Condition0C Short Term, -20C Long Term
SolubilityDMSO
Purity98% by HPLC
SMILES CodeCC(O)=O.O=C([C@@H](NC([C@H](CCCNC(N)=N)NC([C@H](C)NC([C@H](CO)NC([C@@H](NC([C@H](CCCNC(N)=N)NC([C@H](C)NC(CNC([C@H]([C@@H](C)O)NC([C@H](CC(C=C1)=CC=C1F)NC(CNC(CNC([C@H](CC2=CC=CC=C2)N)=O)=O)=O)=O)=O)=O)=O)=O)CCCCN)=O)=O)=O)=O)CCCCN)N
ReferencesBigoni R, et al. Pharmacological characterisation of [[pX]Phe4]nociceptin[1-13]amide analogues. 1. In vitro studies. Naunyn Schmiedebergs Arch Pharmacol. 2002;365[6] 442-449.

More info

[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31. [(pF)Phe4]Nociceptin(1-13)NH2 acetate displays high selectivity over ?, ?, and ? opioid receptors (>3000 fold).