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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $39.10 | Total: $195.50 |
| 1 | 10 | $33.12 | Total: $331.20 |
| 1 | 25 | $28.06 | Total: $701.50 |
| 1 | 50 | $23.92 | Total: $1,196.00 |
| 1 | 100 | $20.70 | Total: $2,070.00 |
Overview
FIDAS-5, a potent and orally active methionine S-adenosyltransferase 2A (MAT2A) inhibitor with an IC50 of 2.1 ?M, competitively inhibits S-adenosylmethionine (SAM) binding to MAT2A. It exhibits anticancer activities.
Chemical Properties
| Molecular Formula | C15H13ClFN |
| Molecular Weight | 261.72 |
| CAS Numbers | 1391934-98-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CNc1ccc(C=Cc2c(F)cccc2Cl)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Zhang W, et al. Fluorinated N,N-dialkylaminostilbenes repress colon cancer by targeting methionine S-adenosyltransferase 2A. ACS Chem Biol. 2013 Apr 19;8[4] 796-803.