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Naltriben mesylate View larger

Naltriben mesylate

AOB5686

CAS: 122517-78-6 (free base: 111555-58-9)

 

Chemical Name: Naltrindole benzofuran mesylate; Naltriben methanesulfonate; (8R-(4bS*,8alpha,8beta,14bbeta))-7-(Cyclopropylmethyl)-6,7,8,14b-tetrahydro-4,8-methano-5H-bisbenzofuro(3,2-e:2',3'-g)isoquinoline-1,8a(9H)-diol

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$21.00

$21.00 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
1100 $9.45 Total: $945.00
150 $10.92 Total: $546.00
125 $12.81 Total: $320.25
110 $15.12 Total: $151.20
15 $17.85 Total: $89.25

Data sheet

Molecular FormulaC26H25NO4.CH3SO3H
Molecular Weight511.59
CAS Numbers122517-78-6
Storage Condition0°C (short term), -20°C (long term), desiccated
SolubilityDMSO
Purity98% by HPLC
SynonymNaltriben methanesulfonate; Naltrindole benzofuran; NTB
IUPAC/Chemical Name17-(Cyclopropylmethyl)-6,7-didehydro-3,14β-dihydroxy-4,5α-epoxy-6,7-2',3'-benzo[b]furanomorphinan mesylate
InChl KeyXRRFZOCDAWPIBB-IDRHMUJXSA-N
InChl CodeInChI=1S/C26H25NO4.CH4O3S/c28-18-8-7-15-11-20-26(29)12-17-16-3-1-2-4-19(16)30-22(17)24-25(26,21(15)23(18)31-24)9-10-27(20)13-14-5-6-14;1-5(2,3)4/h1-4,7-8,14,20,24,28-29H,5-6,9-13H2;1H3,(H,2,3,4)/t20-,24+,25+,26-;/m1./s1
SMILES CodeC[S](O)(=O)=O.[H][C@@]12OC3=C(O)C=CC4=C3[C@@]11CCN(CC3CC3)[C@]([H])(C4)[C@]1(O)CC1=C2OC2=C1C=CC=C2
References1) Miyamoto et al (1993) Involvement of delta2 opioid receptors in the development of mor. dependence in mice. J.Pharmacol.Exp.Ther. 264 1141 PMID: 8383738

2) Portoghese et al (1991) Role of spacer and address components in peptidomimetic δ opioid receptor antagonists related to naltrindole. J.Med.Chem. 34 1715 PMID: 1851846

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