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Enadoline hydrochloride
AOB12923
CAS: 124439-07-2
Chemical Name: 2-(1-Benzofuran-4-yl)-N-methyl-N-[(5R,7S,8S)-7-pyrrolidin-1-yl-1-oxaspiro[4.5]decan-8-yl]acetamide hydrochloride
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 100 | $26.55 | Total: $2,655.00 |
| 1 | 50 | $30.68 | Total: $1,534.00 |
| 1 | 25 | $35.99 | Total: $899.75 |
| 1 | 10 | $42.48 | Total: $424.80 |
| 1 | 5 | $50.15 | Total: $250.75 |
Data sheet
| Molecular Formula | C24H33ClN2O3 |
| Molecular Weight | 432.98 |
| CAS Numbers | 124439-07-2 (HCl), 124378-77-4 (free base) |
| Storage Condition | 0°C (short term), -20°C (long term), desiccated |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| Synonym | Enadoline hydrochloride; Enadoline HCl; ENADOLINE HYDROCHLORIDE; UNII-086I9HO04E; CAM 570; NIH 10672; PD 129290. |
| IUPAC/Chemical Name | 4-Benzofuranacetamide, N-methyl-N-(7-(1-pyrrolidinyl)-1-oxaspiro(4.5)dec-8-yl)-, monohydrochloride, (5R-(5alpha,7alpha,8beta))- |
| InChl Key | ZVVAINSYJGRDTR-TYLGTTGKSA-N |
| InChl Code | InChI=1S/C24H32N2O3.ClH/c1-25(23(27)16-18-6-4-7-22-19(18)9-15-28-22)20-8-11-24(10-5-14-29-24)17-21(20)26-12-2-3-13-26;/h4,6-7,9,15,20-21H,2-3,5,8,10-14,16-17H2,1H3;1H/t20-,21-,24-;/m0./s1 |
| SMILES Code | C1[C@@]2(CC[C@@H]([C@H]1N1CCCC1)N(C(Cc1c3c(occ3)ccc1)=O)C)CCCO2.Cl |
| References | 1) Walsh SL, Strain EC, Abreu ME, Bigelow GE. Enadoline, a selective kappa opioid agonist: comparison with butorphanol and hydromorphone in humans. Psychopharmacology (Berl). 2001 Sep;157(2):151-62. PubMed PMID: 11594439. 2) Walsh SL, Geter-Douglas B, Strain EC, Bigelow GE. Enadoline and butorphanol: evaluation of kappa-agonists on cocaine pharmacodynamics and cocaine self-administration in humans. J Pharmacol Exp Ther. 2001 Oct;299(1):147-58. PubMed PMID: 11561074. |
| PubChem ID | 153555373 |
More info
Novel and selective agonist for the κ-opioid receptor