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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $286.45 | Total: $1,432.25 |
| 1 | 10 | $242.64 | Total: $2,426.40 |
| 1 | 25 | $205.57 | Total: $5,139.25 |
| 1 | 50 | $175.24 | Total: $8,762.00 |
| 1 | 100 | $151.65 | Total: $15,165.01 |
Overview
Patamostat mesylate (E-3123) is a potent protease inhibitor with IC50 values of 39 nM for trypsin, 950 nM for plasmin, and 1.9 ?M for thrombin. This compound demonstrates promising potential in suppressing the pathogenesis and development of acute pancreatitis.
Chemical Properties
| Molecular Formula | C21H24N4O7S2 |
| Molecular Weight | 508.57 |
| CAS Numbers | 114568-32-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C(OC1=CC=C(SCCN2C(=O)CCC2=O)C=C1)C3=CC=C(C=C3)NC(=N)N.O=S(=O)(O)C |
Storage and Handling
0C Short Term, -20C Long Term
References
K Miyamoto, et al. [Effects of E-3123, a New Protease Inhibitor, on Several Protease Activities and on Experimental Acute Pancreatitis]. Nihon Yakurigaku Zasshi. 1988 May;91[5] 285-93.