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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Overview
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
Chemical Properties
| Molecular Formula | C14H19Br2ClN4S |
| Molecular Weight | 470.7 |
| CAS Numbers | 145231-35-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Br.Br.Clc1ccc(CNC(=N)SCCCc2cnc[nH]2)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Mena-Avila E, et al. Clobenpropit, a histamine H3 receptor antagonistinverse agonist, inhibits [3H]-dopamine uptake by human neuroblastoma SH-SY5Y cells and rat brain synaptosomes. Pharmacol Rep. 2018 Feb;70[1] 146-155.