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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $28.05 | Total: $140.25 |
| 1 | 10 | $23.76 | Total: $237.60 |
| 1 | 25 | $20.13 | Total: $503.25 |
| 1 | 50 | $17.16 | Total: $858.00 |
| 1 | 100 | $14.85 | Total: $1,485.00 |
Overview
RAF265 (CHIR-265) (CHIR-265) is a potent selective inhibitor of C-RafB-RafB-Raf V600E with IC50 of 3-60 nM, and exhibits potent inhibition on VEGFR2 phosphorylation with EC50 of 30 nM. Phase 2.
Chemical Properties
| Molecular Formula | C24H16F6N6O |
| Molecular Weight | 518.41 |
| CAS Numbers | 927880-90-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
AACR Meeting Abstracts 2008;2008 4876.