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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $65.45 | Total: $327.25 |
| 1 | 10 | $55.44 | Total: $554.40 |
| 1 | 25 | $46.97 | Total: $1,174.25 |
| 1 | 50 | $40.04 | Total: $2,002.00 |
| 1 | 100 | $34.65 | Total: $3,465.00 |
Overview
AGN 196996 is a potent and selective inhibitor of RAR? (Ki: 2 nM), exhibiting very low affinity for RAR? (Ki: 1087 nM) and RAR? (Ki: 8523 nM).
Chemical Properties
| Molecular Formula | C24H20BrNO5 |
| Molecular Weight | 482.32 |
| CAS Numbers | 958295-17-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCOc1c(Br)cc(cc1C(=O)c1ccc(C)cc1)C(=O)Nc1ccc(cc1)C(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Hammond LA, et al. Antagonists of retinoic acid receptors [RARs] are potent growth inhibitors of prostate carcinoma cells. Br J Cancer. 2001 Aug 3;85[3] 453-62.