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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $102.85 | Total: $514.25 |
| 1 | 10 | $87.12 | Total: $871.20 |
| 1 | 25 | $73.81 | Total: $1,845.25 |
| 1 | 50 | $62.92 | Total: $3,146.00 |
| 1 | 100 | $54.45 | Total: $5,445.00 |
Overview
FMK 9a is an irreversible inhibitor of ATG4B with IC50 values of 80 and 73 nM in the TR-FRET and cellular-based LRA assays.
Chemical Properties
| Molecular Formula | C23H21FN2O3 |
| Molecular Weight | 392.42 |
| CAS Numbers | 1955550-51-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | FCC(=O)CNC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc2ccccc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Qiu Z, et al. Discovery of Fluoromethylketone-Based Peptidomimetics as Covalent ATG4B [Autophagin-1] Inhibitors. ACS Med Chem Lett. 2016 Jun 25;7[8] 802-6.