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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $178.50 | Total: $892.50 |
| 1 | 10 | $151.20 | Total: $1,512.00 |
| 1 | 25 | $128.10 | Total: $3,202.50 |
| 1 | 50 | $109.20 | Total: $5,460.00 |
| 1 | 100 | $94.50 | Total: $9,450.00 |
Overview
SSR240612 is a potent, orally active, specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 nM for B1 receptors and 358-481 nM for B2 receptors, respectively).
Chemical Properties
| Molecular Formula | C42H53ClN4O7S |
| Molecular Weight | 793.41 |
| CAS Numbers | 464930-42-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.COc1ccc2cc(ccc2c1)S(=O)(=O)N[C@H](CC(=O)N[C@H](Cc1ccc(CN2[C@@H](C)CCC[C@H]2C)cc1)C(=O)N(C)C(C)C)c1ccc2OCOc2c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Gougat J, et al. SSR240612 [[2R]-2-[[[3R]-3-[1,3-benzodioxol-5-yl]-3-[[[6-methoxy-2-naphthyl]sulfonyl]amino]propanoyl]amino]-3-[4-[[2R,6S]-2,6-dimethylpiperidinyl]methyl]phenyl]-N-isopropyl-N-methylpropanamide hydrochloride], a new nonpeptide antagonist of the bradykinin B1 receptor biochemical and pharmacological characterization. J Pharmacol Exp Ther. 2004 May;309[2] 661-9.