Donafenib

Donafenib

AT16909

CAS 1130115-44-4

More details

1000 Items

$92.30

$92.30 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $60.35 Total: $301.75
110 $51.12 Total: $511.20
125 $43.31 Total: $1,082.75
150 $36.92 Total: $1,846.00
1100 $31.95 Total: $3,195.00

Overview

Donafenib(Bay 43-9006 (D3)) is a deuterium-labeled Sorafenib which is a multikinase inhibitor(IC50s: 6 nM, 20 nM, and 22 nM for Raf-1, B-Raf, and VEGFR-3, respectively).

Chemical Properties

Molecular FormulaC21H13ClD3F3N4O3
Molecular Weight467.84
CAS Numbers1130115-44-4
SolubilityDMSO
Purity98% by HPLC
SMILES Code[2H]C([2H])([2H])NC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)ccn1

Storage and Handling

0C Short Term, -20C Long Term

References

Wilhelm SM, et al. BAY 43-9006 exhibits broad spectrum oral antitumor activity and targets the RAFMEKERK pathway and receptor tyrosine kinases involved in tumor progression and angiogenesis. Cancer Res. 2004 Oct 1;64[19] 7099-109.