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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $28.05 | Total: $140.25 |
| 1 | 10 | $23.76 | Total: $237.60 |
| 1 | 25 | $20.13 | Total: $503.25 |
| 1 | 50 | $17.16 | Total: $858.00 |
| 1 | 100 | $14.85 | Total: $1,485.00 |
Overview
A-836339 acts as a potent cannabinoid receptor full agonist which has a higher affinity for the peripheral CB2 receptor (Ki = 0.64 nM) over the central CB1 receptor (Ki = 270 nM). It displays analgesic, anti-inflammatory, and anti-hyperalgesic effects in mice.
Chemical Properties
| Molecular Formula | C16H26N2O2S |
| Molecular Weight | 310.45 |
| CAS Numbers | 959746-77-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COCCn1c(C)c(C)sc1=NC(=O)C1C(C)(C)C1(C)C |
Storage and Handling
0C Short Term, -20C Long Term
References
Characterization of a Cannabinoid CB2 Receptor-Selective Agonist, A-836339 [2,2,3,3-Tetramethyl-cyclopropanecarboxylic Acid [3-[2-Methoxy-ethyl]-4,5-dimethyl-3H-thiazol-[2Z]-ylidene]-amide], Using in Vitro Pharmacological Assays, in Vivo Pain Models, and Pharmacological Magnetic Resonance Imaging[J]. Journal of Pharmacology and Experimental Therapeutics, 2009, 328[1] 141-151.