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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $542.30 | Total: $2,711.50 |
| 1 | 10 | $459.36 | Total: $4,593.60 |
| 1 | 25 | $389.18 | Total: $9,729.50 |
| 1 | 50 | $331.76 | Total: $16,588.00 |
| 1 | 100 | $287.10 | Total: $28,710.01 |
Overview
Dirlotapide (CP742033) is an intestinal selective microsomal triglyceride transfer protein (MTP) inhibitor. It reduces body weight in diabetic dogs.Dirlotapide reduces food intake in a dose-dependent manner, possibly by increasing the release of peptide YY into the circulation.
Chemical Properties
| Molecular Formula | C40H33F3N4O3 |
| Molecular Weight | 674.71 |
| CAS Numbers | 481658-94-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(Cc1ccccc1)C(=O)[C@@H](NC(=O)c1cc2cc(NC(=O)c3ccccc3-c3ccc(cc3)C(F)(F)F)ccc2n1C)c1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Wren JA, et al. Biologic activity of dirlotapide, a novel microsomal triglyceride transfer protein inhibitor, for weight loss in obese dogs. J Vet Pharmacol Ther. 2007 Aug;30 Suppl 1 33-42.