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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $49.30 | Total: $246.50 |
| 1 | 10 | $41.76 | Total: $417.60 |
| 1 | 25 | $35.38 | Total: $884.50 |
| 1 | 50 | $30.16 | Total: $1,508.00 |
| 1 | 100 | $26.10 | Total: $2,610.00 |
Overview
AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.
Chemical Properties
| Molecular Formula | C27H32Cl2N2O7 |
| Molecular Weight | 567.46 |
| CAS Numbers | 1003566-93-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CNC(=O)c1cc(Cl)c(OC(C)(C)C(O)=O)cc1OC[C@@H](O)CN1CCC2(Cc3cc(Cl)ccc3O2)CC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Gilchrist A, Gauntner TD, Fazzini A, Alley KM, Pyen DS, Ahn J, Ha SJ, Willett A, Sansom SE, Yarfi JL, Bachovchin KA, Mazzoni MR, Merritt JR. Identifying bias in CCR1 antagonists using radiolabelled binding, receptor internalization, ?-arrestin translocation and chemotaxis assays. Br J Pharmacol. 2014 Nov;171[22] 5127-38. doi 10.1111bph.12835. PubMed PMID 24990525; PubMed Central PMCID PMC4253460.