S1r-in-10

S1r-in-10

AOB14269

1000 Items

$0.00

Overview

Novel selective sigma 1 receptor (S1R) antagonist, exhibiting potent binding affinity for S1R, high selectivity over S2R and 87 other human targets, acceptable in vitro metabolic stability, slowing clearance in liver microsomes, and excellent blood-brain barrier permeability in rats