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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $211.65 | Total: $1,058.25 |
| 1 | 10 | $179.28 | Total: $1,792.80 |
| 1 | 25 | $151.89 | Total: $3,797.25 |
| 1 | 50 | $129.48 | Total: $6,474.00 |
| 1 | 100 | $112.05 | Total: $11,205.00 |
Overview
Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors, and low affinity for dopamine D4, 5-hydroxytryptophan (5-HT2), and ?1-adrenergic receptors.Aplindore Fumarate is used in the study of Parkinson's disease and schizophrenia. Fumarate can be used to study Parkinson's and schizophrenia.
Chemical Properties
| Molecular Formula | C22H22N2O7 |
| Molecular Weight | 426.42 |
| CAS Numbers | 189681-71-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=CC(O)=O)C(O)=O.C(NCC1=CC=CC=C1)[C@@H]2OC=3C4=C(C=CC3OC2)NC(=O)C4 |
Storage and Handling
0C Short Term, -20C Long Term
References
Heinrich JN, et al. Aplindore [DAB-452], a high affinity selective dopamine D2 receptor partial agonist. Eur J Pharmacol. 2006 Dec 15;552[1-3] 36-45.