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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $24.65 | Total: $123.25 |
| 1 | 10 | $20.88 | Total: $208.80 |
| 1 | 25 | $17.69 | Total: $442.25 |
| 1 | 50 | $15.08 | Total: $754.00 |
| 1 | 100 | $13.05 | Total: $1,305.00 |
Overview
Mesdopetam hemitartrate (IRL790 hemitartrate) is an antagonist of dopamine D3 receptor (Ki=90 nM; IC50=9.8 ?M for human recombinant D3 receptor). It has psychomotor stabilizing properties.
Chemical Properties
| Molecular Formula | C28H42F2N2O12S2 |
| Molecular Weight | 700.77 |
| CAS Numbers | 2562346-14-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCNCCOC1=CC(S(=O)(C)=O)=CC(F)=C1.CCCNCCOC2=CC(S(=O)(C)=O)=CC(F)=C2.O=C(O)[C@H](O)[C@@H](O)C(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Waters S, et al. Preclinical Pharmacology of [2-[3-Fluoro-5-Methanesulfonyl-phenoxy]Ethyl][Propyl]amine [IRL790], a Novel Dopamine Transmission Modulator for the Treatment of Motor and Psychiatric Complications in Parkinson Disease. J Pharmacol Exp Ther. 2020;374[1] 113-125.