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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $141.10 | Total: $705.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 100 | $74.70 | Total: $7,470.00 |
Overview
Ecopipam (UNII-0X748O646K) is a potent, selective, and orally active antagonist of dopamine D1D5 receptors, with Kis of 1.2 nM and 2.0 nM, respectively. Ecopipam demonstrates more than 40-fold selectivity over D2, D4, 5-HT, and ?2a receptors (Ki=0.98, 5.52, 0.08, and 0.73 ?M, respectively). It is used in research on schizophrenia and obesity.
Chemical Properties
| Molecular Formula | C19H20ClNO |
| Molecular Weight | 313.82 |
| CAS Numbers | 112108-01-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN1[C@@]2([C@@](C=3C(=CC(Cl)=C(O)C3)CC1)(C=4C(CC2)=CC=CC4)[H])[H] |
Storage and Handling
0C Short Term, -20C Long Term
References
Wu WL, et, al. Dopamine D1D5 receptor antagonists with improved pharmacokinetics design, synthesis, and biological evaluation of phenol bioisosteric analogues of benzazepine D1D5 antagonists. J Med Chem. 2005 Feb 10;48[3] 680-93.