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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $28.05 | Total: $140.25 |
| 1 | 10 | $23.76 | Total: $237.60 |
| 1 | 25 | $20.13 | Total: $503.25 |
| 1 | 50 | $17.16 | Total: $858.00 |
| 1 | 100 | $14.85 | Total: $1,485.00 |
Overview
SIB-1757 (6-methyl-2-[(E)-phenyldiazenyl]pyridin-3) is a selective antagonist of mGlu5 metabotropic glutamate receptor subtype (hmGlu5, IC50 : 0.4 ?M)
Chemical Properties
| Molecular Formula | C12H11N3O |
| Molecular Weight | 213.24 |
| CAS Numbers | 31993-01-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(=NC1=CC=CC=C1)C2=C(O)C=CC(C)=N2 |
Storage and Handling
0C Short Term, -20C Long Term
References
Dogrul A , Ossipov M H , Lai J , et al. Peripheral and spinal antihyperalgesic activity of SIB-1757, a metabotropic glutamate receptor [mGLUR5] antagonist, in experimental neuropathic pain in rats[J]. 2000, 292[2] 0-118.