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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $44.20 | Total: $221.00 |
| 1 | 10 | $37.44 | Total: $374.40 |
| 1 | 25 | $31.72 | Total: $793.00 |
| 1 | 50 | $27.04 | Total: $1,352.00 |
| 1 | 100 | $23.40 | Total: $2,340.00 |
Overview
VU 0469650 is a potent and selective negative allosteric modulator of mGluR1 (IC50 = 99 nM).
Chemical Properties
| Molecular Formula | C22H28N4O |
| Molecular Weight | 364.48 |
| CAS Numbers | 1443748-47-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(=O)(C12CC3CC(C1)CC(C2)C3)N4[C@H](C)CN(CC4)C5=C(C#N)N=CC=C5 |
Storage and Handling
0C Short Term, -20C Long Term
References
Lovell KM, et al. N-Acyl-N'-arylpiperazines as negative allosteric modulators of mGlu1 identification of VU0469650, a potent and selective tool compound with CNS exposure in rats. Bioorg Med Chem Lett. 2013;23[13] 3713-3718.