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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $78.20 | Total: $391.00 |
| 1 | 10 | $66.24 | Total: $662.40 |
| 1 | 25 | $56.12 | Total: $1,403.00 |
| 1 | 50 | $47.84 | Total: $2,392.00 |
| 1 | 100 | $41.40 | Total: $4,140.00 |
Overview
NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA, with an NMDA Ki of 0.85 nM and an NR2B Ca2+ influx IC50 of 9.7 nM.
Chemical Properties
| Molecular Formula | C20H23ClFN3O |
| Molecular Weight | 375.87 |
| CAS Numbers | 700878-19-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cl.Oc1ccc2[nH]c(CN3CCC(Cc4ccccc4F)CC3)nc2c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
McCauley JA, et al. NR2B-selective N-methyl-D-aspartate antagonists synthesis and evaluation of 5-substituted benzimidazoles. J Med Chem. 2004 Apr 8;47[8] 2089-96.