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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $81.60 | Total: $408.00 |
| 1 | 10 | $69.12 | Total: $691.20 |
| 1 | 25 | $58.56 | Total: $1,464.00 |
| 1 | 50 | $49.92 | Total: $2,496.00 |
| 1 | 100 | $43.20 | Total: $4,320.00 |
Overview
JNJ-61432059 is an orally active and selective negative modulator of TARP ?-8 selective AMPAR (pIC50: 9.7).
Chemical Properties
| Molecular Formula | C25H22FN5O2 |
| Molecular Weight | 443.47 |
| CAS Numbers | 2035814-50-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OC1CCN(CC1)c1nccc2c(c(nn12)-c1ccc(F)cc1)-c1ccc2NC(=O)Cc2c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Savall BM, et al. Discovery of Imidazo[1,2-a]pyrazines and Pyrazolo[1,5-c]pyrimidines as TARP ?-8 Selective AMPAR Negative Modulators. ACS Med Chem Lett. 2018 Dec 26;10[3] 267-272.